Preface.

1 Overview of Drug Transporter Families (Guofeng You and Marilyn E. Morris).

2 Organic Cation Transporters (Thomas J. Urban and Kathleen M. Giacomini).

3 Organic Cation/Carnitine Transporters (Ijaz A. Qureshi, Ihsan Elimrani, Ernest Seidman, and Grant Mitchell).

4 Organic Anion Transporters (Megha Nagle, David M. Truong, Vibha Bhatnagar, Gregory Kaler, Kevin T. Bush, Wei Wu, Satish A. Eraly, and Sanjay K. Nigam).

5 Organic Anion–Transporting Polypeptides (Rommel G. Tirona and Richard B. Kim).

6 Mammalian Oligopeptide Transporters (Stephen M. Carl, Dea Herrera-Ruiz, Rajinder K. Bhardwaj, Olafur Gudmundsson, and Gregory T. Knipp).

7 Monocarboxylate Transporters (Justin A. Spanier and Lester R. Drewes).

8 Nucleoside Transporters: CNTs and ENTs (Li Xia, Mingyan Zhou, and Joanne Wang).

9 Bile Acid Transporters (Jyrki J. Eloranta and Gerd A. Kullak-Ublick).

10 Multidrug Resistance Protein: P-Glycoprotein (Frances J. Sharom).

11 Multidrug Resistance Proteins of the ABCC Subfamily (Anne T. Nies, Maria Rius, and Dietrich Keppler).

12 Breast Cancer Resistance Protein (Robert W. Robey, Orsolya Polgar, John Deeken, Kenneth K. W. To, and Susan E. Bates).

13 Drug Transport in the Liver (Pieter Annaert, Brandon Swift, Jin Kyung Lee, and Kim L. R. Brouwer).

14 Drug Transport in the Brain (Patrick T. Ronaldson, Karlo Babakhanian, and Reina Bendayan).

15 Drug Transport in the Kidney (Naohiko Anzai and Hitoshi Endou).

16 Drug Transporters in the Intestine (Yaming Su and Patrick J. Sinko).

17 Regulation of Drug Transporter Activity (Mei Hong and Guofeng You).

18 Experimental Approaches to the Study of Drug Transporters (Yoshiyuki Kubo, Yukio Kato, and Akira Tsuji).

19 In Vitro–In Vivo Scale-up of Drug Transport Activities (Kazuya Maeda and Yuichi Sugiyama).

20 Age- and Gender-Related Differences in Xenobiotic Transporter Expression (Curtis D. Klaassen and Xingguo Cheng).

21 Polymorphisms of Drug Transporters and Clinical Relevance (Leslie W. Chinn, Jason M. Gow, and Deanna L. Kroetz).

22 Diet/Nutrient Interactions with Drug Transporters (Xiaodong Wang and Marilyn E. Morris).

23 Interplay of Drug Transporters and Enzymes on Hepatic Drug Processing (K. Sandy Pang, Huadong Sun, and Shanjun Liu).

24 Clinical Relevance: Drug–Drug Interactions, Pharmacokinetics, Pharmacodynamics, and Toxicity (Serena Marchetti, Roberto Mazzanti, Jos H. Beijnen, and Jan H. M. Schellens).

Index.